Palladium-catalyzed cascade allylation/carbopalladation/cross coupling: A novel three-component reaction for the synthesis of 3,3-disubstituted-2,3- dihydrobenzofurans

Magali Szlosek-Pinaud, Philippe Diaz, Jean Martinez, Frédéric Lamaty

Research output: Contribution to journalArticlepeer-review

Abstract

A novel one-pot palladium-catalyzed cascade between 2-iodophenol, methyl bromomethylacrylate and an arylboronic acid provides an efficient access to heterocycles possessing the 3,3-disubstituted-2,3-dihydrobenzofuran skeleton via allylation/carbopalladation/Suzuki cross-coupling.

Original languageEnglish
Pages (from-to)8657-8659
Number of pages3
JournalTetrahedron Letters
Volume44
Issue number48
DOIs
StatePublished - Nov 24 2003

Keywords

  • Catalysis
  • Cyclization
  • Multicomponent reactions
  • Oxygen heterocycles
  • Palladium

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