Abstract
The reaction of hippuric acid with trifluoroacetic anhydride in the presence of cyclopentadiene affords useful bicyclic α-amino acid derivatives bearing β-trifluoroacetoxy and β-trifluoromethyl groups.
Original language | English |
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Pages (from-to) | 101-102 |
Number of pages | 2 |
Journal | Synlett |
Volume | 1995 |
Issue number | 1 |
DOIs | |
State | Published - Jan 1995 |
Keywords
- 2-phenyl-5-oxazolone
- Dakin-West reaction
- Diels-Alder cycloaddition
- tandem sequence
- β-trifluoromethyl α-amino acids