Synthesis of bridged bicyclic β-trifluoroacetoxy β-trifluoromethyl α-amino acid derivatives by an original dakin-west/Diels-Alder tandem sequence

Thierry Cufos; Philippe Diaz; Lucien Stella

doi:10.1055/s-1995-4844

Synthesis of bridged bicyclic β-trifluoroacetoxy β-trifluoromethyl α-amino acid derivatives by an original dakin-west/Diels-Alder tandem sequence

Thierry Cufos
, Philippe Diaz
, Lucien Stella

Aix-Marseille Université

Research output: Contribution to journal › Article › peer-review

5 Scopus citations

Abstract

The reaction of hippuric acid with trifluoroacetic anhydride in the presence of cyclopentadiene affords useful bicyclic α-amino acid derivatives bearing β-trifluoroacetoxy and β-trifluoromethyl groups.

Original language	English
Pages (from-to)	101-102
Number of pages	2
Journal	Synlett
Volume	1995
Issue number	1
DOIs	https://doi.org/10.1055/s-1995-4844
State	Published - Jan 1995

Keywords

2-phenyl-5-oxazolone
Dakin-West reaction
Diels-Alder cycloaddition
tandem sequence
β-trifluoromethyl α-amino acids

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10.1055/s-1995-4844

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title = "Synthesis of bridged bicyclic β-trifluoroacetoxy β-trifluoromethyl α-amino acid derivatives by an original dakin-west/Diels-Alder tandem sequence",

abstract = "The reaction of hippuric acid with trifluoroacetic anhydride in the presence of cyclopentadiene affords useful bicyclic α-amino acid derivatives bearing β-trifluoroacetoxy and β-trifluoromethyl groups.",

keywords = "2-phenyl-5-oxazolone, Dakin-West reaction, Diels-Alder cycloaddition, tandem sequence, β-trifluoromethyl α-amino acids",

author = "Thierry Cufos and Philippe Diaz and Lucien Stella",

year = "1995",

month = jan,

doi = "10.1055/s-1995-4844",

language = "English",

volume = "1995",

pages = "101--102",

journal = "Synlett",

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T1 - Synthesis of bridged bicyclic β-trifluoroacetoxy β-trifluoromethyl α-amino acid derivatives by an original dakin-west/Diels-Alder tandem sequence

AU - Cufos, Thierry

AU - Diaz, Philippe

AU - Stella, Lucien

PY - 1995/1

Y1 - 1995/1

N2 - The reaction of hippuric acid with trifluoroacetic anhydride in the presence of cyclopentadiene affords useful bicyclic α-amino acid derivatives bearing β-trifluoroacetoxy and β-trifluoromethyl groups.

AB - The reaction of hippuric acid with trifluoroacetic anhydride in the presence of cyclopentadiene affords useful bicyclic α-amino acid derivatives bearing β-trifluoroacetoxy and β-trifluoromethyl groups.

KW - 2-phenyl-5-oxazolone

KW - Dakin-West reaction

KW - Diels-Alder cycloaddition

KW - tandem sequence

KW - β-trifluoromethyl α-amino acids

UR - https://www.scopus.com/pages/publications/0002408051

U2 - 10.1055/s-1995-4844

DO - 10.1055/s-1995-4844

M3 - Article

AN - SCOPUS:0002408051

SN - 0936-5214

VL - 1995

SP - 101

EP - 102

JO - Synlett

JF - Synlett

IS - 1

ER -

Synthesis of bridged bicyclic β-trifluoroacetoxy β-trifluoromethyl α-amino acid derivatives by an original dakin-west/Diels-Alder tandem sequence

Abstract

Keywords

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